主な投稿論文

  • TOP  >  
  • 主な投稿論文

Achievements主な投稿論文

  • Upregulation of long non‑coding RNA LINC00460 in EGFR‑mutant lung cancer indicates a poor prognosis in patients treated with osimertinib
    著者
    Nakano, Yuta., Isobe, Kazutoshi., Yoshizawa, Takahiro., Urabe, Naohisa., Homma, Sakae., Kishi, Kazuma.
    雑誌名
    Onco Lett
    26
    ページ
    380
    2023
    DOI
    10.3892/ol.2023.13966
    PMID
    37559586
    Online published
    2023 Jul 20
  • Trastuzumab deruxtecan in metastatic breast cancer with variable HER2 expression: the phase 2 DAISY trial
    著者
    Mosele, Fernanda., Deluche, Elise., Lusque, Amelie., Le Bescond, Loïc., Filleron, Thomas., Pradat, Yoann., Ducoulombier, Agnes., Pistilli, Barbara., Bachelot, Thomas., Viret, Frederic., Levy, Christelle., Signolle, Nicolas., Alfaro, Alexia., T. N. Tran, Diep., Judith Garberis, Ingrid., Talbot, Hugues., Christodoulidis, Stergios., Vakalopoulou, Maria., Droin, Nathalie., Stourm, Aurelie., Kobayashi, Maki., Kakegawa, Tomoya., Lacroix, Ludovic., Saulnier, Patrick., Job, Bastien., Deloger, Marc., Jimenez, Marta., Mahier, Celine., Baris, Vianney., Laplante, Pierre., Kannouche, Patricia., Marty, Virginie., Lacroix-Triki, Magali., Diéras, Veronique., André, Fabrice.
    雑誌名
    Nat Med
    29
    ページ
    2110-2120
    2023
    DOI
    10.1038/s41591-023-02478-2
    PMID
    37488289
    Online published
    2023 Jul 24
  • Evaluation of control of additive concentration in gradient analysis of supercritical fluid chromatography-coupled to tandem mass spectrometry
    著者
    Yamaguchi, Mayu., Tsuji, Makoto.
    雑誌名
    J Chromatogr A
    1705
    ページ
    464193
    2023
    DOI
    10.1016/j.chroma.2023.464193
    PMID
    37429077
    Online published
    2023 Jul 02
  • N-Aryl Indoles as a Novel Class of Potent NaV1.7 Inhibitors
    著者
    Karanjule, Narayan., Hayashi, Noriyuki., Suzuki, Sayaka., Tsuda, Toshifumi., Tokumaru, Eri., Tanaka, Kyosuke., Kimoto, Hiroko., Domon, Yuki., Takahashi, Sakiko., Kubota, Kazufumi., Kitano, Yutaka., Yokoyama, Tomihisa., Koishi, Ryuta., Fujiwara, Chie., Inaba, Shinichi., Asano, Daigo., Sakakura, Tomoko., Takasuna, Kiyoshi., Shinozuka, Tsuyoshi.
    雑誌名
    ACS Med Chem Lett
    14
    ページ
    788-793
    2023
    DOI
    10.1021/acsmedchemlett.3c00079
    PMID
    37312847
    Online published
    2023 Jun 08
  • Deep learning generates custom-made logistic regression models for explaining how breast cancer subtypes are classified
    著者
    Shibahara, Takuma., Wada, Chisa., Yamashita, Yasuho., Fujita, Kazuhiro., Sato, Masamichi., Kuwata, Junichi., Okamoto, Atsushi., Ono, Yoshimasa.
    雑誌名
    PLoS One
    18
    ページ
    e0286072
    2023
    DOI
    10.1371/journal.pone.0286072
    PMID
    37216350
    Online published
    2023 May 22
  • Neuroprotection and axon regeneration by novel low-molecular-weight compounds through the modification of DOCK3 conformation
    著者
    Namekata, Kazuhiko., Tsuji, Naoki., Guo, Xiaoli., Nishijima, Euido., Honda, Sari., Kitamura, Yuta., Yamasaki, Atsushi., Kishida, Masamichi., Takeyama, Jun., Ishikawa, Hirokazu., Shinozaki, Youichi., Kimura, Atsuko., Harada, Chikako., Harada, Takayuki.
    雑誌名
    Cell Death Discov
    9
    ページ
    166
    2023
    DOI
    10.1038/s41420-023-01460-8
    PMID
    37188749
    Online published
    2023 May 15
  • Blood glucose trends in glycogen storage disease type Ia: A cross-sectional study
    著者
    Fukuda,Tokiko., Ito, Tetsuya., Hamazaki, Takashi., Inui, Ayano., Ishige, Mika., Kagawa, Reiko., Sakai, Norio., Watanabe, Yoriko., Kobayashi, Hironori., Wasaki, Yosuke., Taura, Junki., Imamura, Yuki., Tsukiuda, Tsutomu., Nakamura, Kimitoshi.
    雑誌名
    J Inherit Metab Dis
    46
    ページ
    618-633
    2023
    DOI
    10.1002/jimd.12610
    PMID
    37114839
    Online published
    2023 Apr 28
  • Suppression of TDP-43 aggregation by artificial peptide binder targeting to its low complexity domain
    著者
    Kamagata, Kiyoto., Kanbayashi, Saori., Koda, Shuichi., Kadotani, Akito., Ubukata, Osamu., Tashima, Takumi.
    雑誌名
    Biochem Biophys Res Commun
    662
    ページ
    119-125
    2023
    DOI
    10.1016/j.bbrc.2023.04.064
    PMID
    37104882
    Online published
    2023 Apr 20
  • Recognition mechanism of a novel gabapentinoid drug, mirogabalin, for recombinant human α2δ1, a voltage-gated calcium channel subunit
    著者
    Kozai, Daisuke., Numoto, Nobutaka., Nishikawa, Kouki., Kamegawa, Akiko., Kawasaki, Shohei., Hiroaki, Yoko., Irie, Katsumasa., Oshima, Atsunori., Hanzawa, Hiroyuki., Shimada , Kousei., Kitano, Yutaka., Fujiyoshi, Yoshinori.
    雑誌名
    J Mol Biol
    435
    ページ
    168049
    2023
    DOI
    10.1016/j.jmb.2023.168049
    PMID
    36933823
    Online published
    2023 Mar 17
  • A novel Menin-MLL1 inhibitor, DS-1594a, prevents the progression of acute leukemia with rearranged MLL1 or mutated NPM1
    著者
    Numata, Masashi., Haginoya, Noriyasu., Shiroishi, Machiko., Hirata, Tsuyoshi., Sato-Otsubo, Aiko., Yoshikawa, Kenji., Takata, Yoshimi., Nagase, Reina., Kashimoto, Yoshinori., Suzuki, Makoto., Schulte, Nina., Polier, Gernot., Kurimoto, Akiko., Tomoe, Yumiko., Toyota, Akiko., Yoneyama, Tomoko., Imai, Emi., Watanab, Kenji., Hamada, Tomoaki., Kanada, Ryutaro., Watanabe, Jun., Kagoshima, Yoshiko., Tokumaru, Eri., Murata, Kenji., Baba, Takayuki., Shinozaki, Taeko., Ohtsuka, Masami., Goto, Koichi., Karibe, Tsuyoshi., Deguchi, Takao., Gocho, Yoshihiro., Yoshida, Masanori., Tomizawa, Daisuke., Kato, Motohiro., Tsutsumi, Shinji., Kitagawa, Mayumi., Abe, Yuki.
    雑誌名
    Cancer Cell Int
    23
    ページ
    36
    2023
    DOI
    10.1186/s12935-023-02877-y
    PMID
    36841758
    Online published
    2023 Feb 25
  • Changes in HER3 expression profiles between primary and recurrent gynecological cancers
    著者
    Kojima,Yuki., Sudo, Kazuki., Yoshida, Hiroshi., Yazaki, Shu., Tokura, Momoko., Mizoguchi, Chiharu., Okuma S, Hitomi., Kita, Shosuke., Yamamoto, Kasumi., Nishikawa, Tadaaki., Noguchi, Emi., Shimoi, Tatsunori., Tanase, Yasuhito., Uno, Masaya., Ishikawa, Mitsuya., Kato, Tomoyasu., Koyama, Kumiko., Kobayashi, Maki., Kakegawa, Tomoya., Fujiwara, Yasuhiro., Yonemori, Kan.
    雑誌名
    Cancer Cell Int
    23
    ページ
    18
    2023
    DOI
    10.1186/s12935-022-02844-z
    PMID
    36737733
    Online published
    2023 Feb 03
  • Selection of the methylotrophic yeast Ogataea minuta as a high-producing host for heterologous protein expression
    著者
    Tsuda, Masashi., Nakatani, Yuki., Baba, Satoshi., Tanaka, Isshin., Ichikawa, Kimihisa., Nonaka, Koichi., Ito, Rie., Yoko-O, Takehiko., Chiba Yasunori.
    雑誌名
    J Biosci Bioeng
    135
    ページ
    196-202
    2023
    DOI
    10.1016/j.jbiosc.2022.12.006
    PMID
    36702678
    Online published
    2023 Jan 24
  • Discovery of a novel ATP-competitive MEK inhibitor DS03090629 that overcomes resistance conferred by BRAF overexpression in BRAF-mutated melanoma
    著者
    Takano, Kohei., Munehira, Yoichi., Hatanaka, Mana., Murakami, Ryo., Shibata, Yoshihiro., Shida, Takeshi., Takeuchi, Kosuke., Takechi, Sho., Tabata, Toshiki., Shimada, Takashi., Kishikawa, Shuhei., Matsui, Yumi., Ubukata, Osamu., Seki, Takahiko., Kaneta, Yasuyuki.
    雑誌名
    Mol Cancer Ther
    22
    ページ
    317-332
    2023
    DOI
    10.1158/1535-7163.MCT-22-0306
    PMID
    36622773
    Online published
    2023 Jan 09
  • Discovery of DS-9300: A Highly Potent, Selective, and Once-Daily Oral EP300/CBP Histone Acetyltransferase Inhibitor
    著者
    Kanada, Ryutaro., Kagoshima, Yoshiko., Suzuki, Takashi., Nakamura, Akifumi., Funami, Hideaki., Watanabe, Jun., Asano, Masayoshi., Takahashi, Mizuki., Ubukata, Osamu., Suzuki, Kanae., Aikawa, Tomoya., Sato, Kazumi., Goto, Megumi., Setsu, Genzui., Ito, Kentaro., Kihara, Kawori., Kuroha, Mutsumi., Kohno, Takashi., Ogiwara, Hideaki., Isoyama, Takeshi., Tominaga, Yuichi., Higuchi, Saito., Naito, Hiroyuki.
    雑誌名
    J Med Chem
    66
    ページ
    695-715
    2023
    DOI
    10.1021/acs.jmedchem.2c01641
    PMID
    36572866
    Online published
    2022 Dec 26
  • Inhibition of Liquid–Liquid Phase Separation for Breaking the Solubility Barrier of Amorphous Solid Dispersions to Improve Oral Absorption of Naftopidil
    著者
    Fukiage, Masafumi., Suzuki, Kyosuke., Matsuda, Maki., Nishida, Yohei., Oikawa, Michinori., Fujita, Takuya., Kawakami, Kohsaku.
    雑誌名
    Pharmaceutics
    14
    ページ
    2664
    2022
    DOI
    10.3390/pharmaceutics14122664
    PMID
    36559158
    Online published
    2022 Nov 30
  • Practical Synthetic Method of Ogipeptin Derivatives
    著者
    Takiguchi, Shingo., Nishi, Takahide.
    雑誌名
    Synlett
    34
    ページ
    277-282
    2023
    DOI
    10.1055/a-1981-4379
    PMID
    Online published
    2022 Nov 17
  • Inflammation of the cardiac coronary artery in ICR mice
    著者
    Yasuno,Kyohei., Imaoka, Masako., Ohsawa, Tetsuya., Okado, Keiko., Kai, Kiyonori., Tsuchiya, Yoshimi.
    雑誌名
    J Toxicol Pathol
    35
    ページ
    345-348
    2022
    DOI
    10.1293/tox.2022-0022
    PMID
    36406175
    Online published
    2022 Jun 11
  • Identification and characterization of lysophosphatidylcholine 14:0 as a biomarker for drug-induced lung disease
    著者
    Saito, Kosuke., Gemma, Akihiko., Tatsumi, Koichiro., Hattori, Noboru., Ushiki, Atsuhito., Tsushima, Kenji., Saito, Yoshinobu., Abe, Mitsuhiro., Horimasu, Yasushi., Kashiwada, Takeru., Mori, Kazuhiko., Sato, Motonobu., Nishiya, Takayoshi., Takamatsu, Kazuhiko., Sun, Yuchen., Arakawa, Noriaki., Izumi, Takashi., Ohno, Yasuo., Saito, Yoshiro., Hanaoka, Masayuki.
    雑誌名
    Sci Rep
    12
    ページ
    19819
    2022
    DOI
    10.1038/s41598-022-24406-z
    PMID
    36396675
    Online published
    2022 Nov 17
  • Novel Antibody Exerts Antitumor Effect through Downregulation of CD147 and Activation of Multiple Stress Signals
    著者
    Fukuchi, Keisuke., Nanai, Kayoko., Yuita, Hiroshi., Maru, Chikako., Tsukada, Jun., Ishigami, Masato., Nagai, Yoko., Nakano, Yoko., Yoshimura, Chigusa., Yoneda, Kozo., Amano, Masato., Nakamura, Kensuke., Oda, Yoko., Nishigohri, Haruyuki., Yamamoto, Shoji., Ohnishi-Totoki, Yusuke., Inaki, Koichiro., Komori, Hironobu., Nakano, Rika., Kanari, Yoshiyuki., Nishida, Atsuko., Matsui, Yumi., Funo, Satoko., Takahashi, Sayako., Ohtsuka, Toshiaki., Agatsuma, Toshinori.
    雑誌名
    J Oncol
    2022
    ページ
    3552793
    2022
    DOI
    10.1155/2022/3552793
    PMID
    36385956
    Online published
    2022 Nov 04
  • Spatial and Quantitative Analysis of Tumor-Associated Macrophages: Intratumoral CD163-/PD-L1+ TAMs as a Marker of Favorable Clinical Outcomes in Triple-Negative Breast Cancer
    著者
    Shinohara, Hajime., Kobayashi, Maki., Hayashi, Kumiko., Nogawa, Daichi., Asakawa, Ayaka., Ohata, Yae., Kubota, Kazuishi., Takahashi, Hisashi., Yamada, Miyuki., Tokunaga, Masanori., Kinugasa, Yusuke., Oda, Goshi., Nakagawa, Tsuyoshi., Onishi, Iichiroh., Kinowaki, Yuko., Kurata, Morito., Ohashi, Kenichi., Kitagawa, Masanobu., Yamamoto, Kouhei.
    雑誌名
    Int J Mol Sci
    23
    ページ
    13235
    2022
    DOI
    10.3390/ijms232113235
    PMID
    36362023
    Online published
    2022 Oct 31
  • The Novel Gabapentinoid Mirogabalin Prevents Upregulation of α2δ-1 Subunit of Voltage-Gated Calcium Channels in Spinal Dorsal Horn in a Rat Model of Spinal Nerve Ligation
    著者
    Domon,Yuki., Kobayashi, Naoko., Kubota, Kazufumi., Kitano, Yutaka., Ueki, Hideaki., Shimojo, Yumiko., Ishikawa, Kayoko., Ofune, Yuka.
    雑誌名
    Drug Res (Stuttg)
    73
    ページ
    54-60
    2022
    DOI
    10.1055/a-1941-8907
    PMID
    36216339
    Online published
    2022 Oct 10
  • Stratifin as a novel diagnostic biomarker in serum for diffuse alveolar damage
    著者
    Arakawa,Noriaki., Ushiki, Atsuhito., Abe, Mitsuhiro., Matsuyama, Shinichiro., Saito, Yoshinobu., Kashiwada, Takeru., Horimasu, Yasushi., Gemma, Akihiko., Tatsumi, Koichiro., Hattori, Noboru., Tsushima, Kenji., Miyashita, Keiko., Saito, Kosuke., Nakamura, Ryosuke., Toyoda, Takeshi., Ogawa, Kumiko., Sato, Motonobu., Takamatsu, Kazuhiko., Mori, Kazuhiko., Nishiya, Takayoshi., Izumi, Takashi., Ohno, Yasuo., Saito, Yoshiro., Hanaoka, Masayuki.
    雑誌名
    Nat Commun
    13
    ページ
    5854
    2022
    DOI
    10.1038/s41467-022-33160-9
    PMID
    36195613
    Online published
    2022 Oct 04
  • Effect of Trastuzumab Deruxtecan on QT/QTc Interval and Pharmacokinetics in HER2-Positive or HER2-Low Metastatic/Unresectable Breast Cance
    著者
    Shimomura, Akihiko., Takano, Toshimi., Takahashi, Shunji., Sagara, Yasuaki., Watanabe, Junichiro., Tokunaga, Eriko., Shinkai, Tetsu., Kamio, Takahiro., Kikumori, Kunika., Kamiyama, Emi., Fujisaki, Yoshihiko., Saotome, Dan., Yamashita, Toshinari.
    雑誌名
    Clin Pharmacol Ther
    113
    ページ
    160-169
    2023
    DOI
    10.1002/cpt.2757
    PMID
    36164935
    Online published
    2022 Sep 27
  • Quantitative high-throughput analysis of tumor infiltrating lymphocytes in breast cancer
    著者
    Hayashi, Kumiko., Nogawa, Daichi., Kobayashi, Maki., Asakawa, Ayaka., Ohata, Yae., Kitagawa, Shota., Kubota, Kazuishi., Takahashi, Hisashi., Yamada, Miyuki., Oda, Goshi., Nakagawa, Tsuyoshi., Uetake, Hiroyuki., Onishi, Iichiroh., Kinowaki, Yuko., Kurata, Morito., Kitagawa, Masanobu., Yamamoto, Kouhei.
    雑誌名
    Front Oncol
    12
    ページ
    901591
    2022
    DOI
    10.3389/fonc.2022.901591
    PMID
    36132149
    Online published
    2022 Sep 05
  • Pan-cancer gene expression analysis of tissue microarray using EdgeSeq oncology biomarker panel and a cross-comparison with HER2 and HER3 immunohistochemical analysis
    著者
    Inaki,Koichiro., Shibutani, Tomoko., Maeda, Naoyuki., Eppenberger-Castori, Serenella., Nicolet, Stefan., Kaneda, Yuki., Koyama, Kumiko., Qiu, Yang., Wakita, Kenichi., Murakami, Masato.
    雑誌名
    PLoS One
    17
    ページ
    e027414
    2022
    DOI
    10.1371/journal.pone.0274140
    PMID
    36137139
    Online published
    2022 Sep 22
  • Potent and selective PTDSS1 inhibitors induce collateral lethality in cancers with PTDSS2 deletion
    著者
    Yoshihama,Yohei., Namiki, Hidenori., Kato, Taiga., Shimazaki, Naomi., Takaishi, Sachiko., Kadoshima-Yamaoka, Kumiko., Yukinaga, Hideo., Maeda, Naoyuki., Shibutani, Tomoko., Fujimoto, Kazunori., Hirasawa, Makoto., Goto, Hiroki., Wada, Naoya., Tsutsumi, Shinji., Hirota, Yasuhide., Ishikawa, Tomoki., Yamamoto, Shoji.
    雑誌名
    Cancer Res
    82
    ページ
    4031-4043
    2022
    DOI
    10.1158/0008-5472.CAN-22-1006
    PMID
    36054550
    Online published
    2022 Sep 02
  • Identification and characterization of a novel thermo-stable endo-β-N-acetylglucosaminidase from Rhizomucorpusillus
    著者
    Nishizawa, Hanako., Iwamoto, Mitsuhiro., Ono, Yasunori.
    雑誌名
    J Biosci Bioeng
    134
    ページ
    295-300
    2022
    DOI
    10.1016/j.jbiosc.2022.06.013
    PMID
    35961816
    Online published
    2022 Aug 10
  • Novel protein kinase cAMP-Activated Catalytic Subunit Alpha (PRKACA) inhibitor shows anti-tumor activity in a fibrolamellar hepatocellular carcinoma model
    著者
    Toyota, Akiko., Goto, Megumi., Miyamoto, Masaya., Nagashima, Yoko., Iwasaki, Shiho., Komatsu, Takahiro., Momose, Takayuki., Yoshida, Keisuke., Tsukada, Tomoharu., Matsufuji, Tetsuyoshi., Ohno, Ami., Suzuki, Makoto., Ubukata, Osamu., Kaneta, Yasuyuki.
    雑誌名
    Biochem Biophys Res Commun
    621
    ページ
    157-161
    2022
    DOI
    10.1016/j.bbrc.2022.07.008
    PMID
    35839742
    Online published
    2022 Jul 07
  • Impact of the Clinical Trials Act 2018 on clinical trial activity in Japan from 2018 to 2020: a retrospective database study using new and conventional Japanese registries
    著者
    Taruno, Hiroyuki., Oba, Mari S., Takizawa, Osamu., Kikuchi, Kayoko., Matsui, Kazuaki., Shikano, Mayumi.
    雑誌名
    BMJ Open
    12
    ページ
    e059092
    2022
    DOI
    10.1136/bmjopen-2021-059092
    PMID
    35851007
    Online published
    2022 Jul 18
  • Total Synthesis and Structural Elucidation of Ogipeptins
    著者
    Takiguchi, Shingo., Hirota-Takahata,Yuki., Nishi, Takahide.
    雑誌名
    Org Lett
    24
    ページ
    4935-4938
    2022
    DOI
    10.1021/acs.orglett.2c01863
    PMID
    35796660
    Online published
    2022 Jul 07
  • Systematic Exploration of Passive Permeability in Tetrapeptides with Hydrogen­­–Bond Accepting Amino Acid Side Chains
    著者
    Shimizu, Hiroki., Renslo, Adam.
    雑誌名
    ChemMedChem
    17
    ページ
    e202200204
    2022
    DOI
    10.1002/cmdc.202200204
    PMID
    35696654
    Online published
    2022 Jun 13
  • Microarray-based gene expression analysis combined with laser capture microdissection is beneficial in investigating the modes of action of ocular toxicity
    著者
    Shirai, Makoto., Niino, Noriyo., Mori, Kazuhiko., Kai, Kiyonori.
    雑誌名
    J Toxicol Pathol
    35
    ページ
    171-182
    2022
    DOI
    10.1293/tox.2021-0064
    PMID
    35516843
    Online published
    2021 Dec 18
  • Patritumab deruxtecan (HER3-DXd), a novel HER3 directed antibody drug conjugate, exhibits in vitro activity against breast cancer cells expressing HER3 mutations with and without HER2 overexpression
    著者
    Koyama ,Kumiko., Ishikawa, Hirokazu., Abe, Manabu., Shiose, Yoshinobu., Ueno, Suguru., Qiu, Yang., Nakamaru, Kenji., Murakami, Masato.
    雑誌名
    PLoS One.
    17
    ページ
    e0267027
    2022
    DOI
    10.1371/journal.pone.0267027
    PMID
    35503762
    Online published
    2022 May 03
  • Determination of key residues in MRGPRX2 to enhance pseudo-allergic reactions induced by fluoroquinolones
    著者
    Hamamura-Yasuno, Eri., Matsushita, Junya., Sato, Seiji., Shimada, Takashi., Tsuchiya, Yoshimi., Fujimoto, Kazunori., Mori, Kazuhiko.
    雑誌名
    Sci Rep.
    12
    ページ
    6650
    2022
    DOI
    10.1038/s41598-022-10549-6.
    PMID
    35459883
    Online published
    2022 Apr 22
  • Application of the advanced Marfey’s method for the determination of the absolute configuration of ogipeptins
    著者
    Takiguchi, Shingo., Hirota-Takahata, Yuki., Nishi, Takahide.
    雑誌名
    Tetrahedron Letters
    96
    ページ
    153760
    2022
    DOI
    10.1016/j.tetlet.2022.153760
    PMID
    Online published
    2022 Mar 30
  • Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring
    著者
    Kanada, Ryutaro., Kagoshima, Yoshiko., Asano, Masayoshi., Suzuki, Takashi., Murata, Takeshi., Haruta, Makoto., Takahashi, Mizuki., Ubukata, Osamu., Hashimoto, Kazuyuki., Obata, Kenichi., Kihara, Kawori., Kuroha, Mutsumi., Banjo, Toshihiro., Togashi, Noriko., Sato, Kazumi., Yamamoto, Yuka., Suzuki, Kanae., Isoyama, Takeshi., Tominaga, Yuichi., Higuchi, Saito., Naito, Hiroyuki.
    雑誌名
    Bioorg Med Chem Lett
    66
    ページ
    128726
    2022
    DOI
    10.1016/j.bmcl.2022.128726
    PMID
    3541341
    Online published
    2022 Apr 09
  • CYP2C8-Mediated Formation of a Human Disproportionate Metabolite of the Selective Na V 1.7 Inhibitor DS-1971a, a Mixed Cytochrome P450 and Aldehyde Oxidase Substrate
    著者
    Asano, Daigo., Hamaue, Syoya., Zahir, Hamim., Shiozawa, Hideyuki ., Nishiya, Yumi., Kimura, Takako., Kazui, Miho., Yamamura, Naotoshi., Ikeguchi, Marie., Shibayama, Takahiro., Inoue, Shin-Ichi., Shinozuka, Tsuyoshi., Watanabe, Toshiyuki., Yahara, Chizuko., Watanabe, Nobuaki., Yoshinari, Kouichi.
    雑誌名
    Drug Metab Dispos
    50
    ページ
    235-242
    2022
    DOI
    10.1124/dmd.121.000665
    PMID
    34930785
    Online published
    2021 Dec 20
  • DS-7300a, a DNA Topoisomerase I Inhibitor, DXd-based Antibody-Drug Conjugate Targeting B7-H3 Exerts Potent Antitumor Activities in Preclinical Models
    著者
    Yamato,Michiko., Hasegawa, Jun., Maejima, Takanori., Hattori, Chiharu., Kumagai, Kazuyoshi., Watanabe, Akiko., Nishiya, Yumi., Shibutani, Tomoko., Aida, Tetsuo., Hayakawa, Ichiro., Nakada, Takashi., Abe, Yuki., Agatsuma, Toshinori.
    雑誌名
    Mol Cancer Ther
    21
    ページ
    635-646
    2022
    DOI
    10.1158/1535-7163.MCT-21-0554
    PMID
    35149548
    Online published
    2022 Feb 11
  • A gut-derived metabolite alters brain activity and anxiety behaviour in mice
    著者
    Needham, Brittany D., Funabashi, Masanori., Adame, Mark D., Wang, Zhuo., Boktor, Joseph C., Haney, Jillian., Wu, Wei-Li., Rabut, Claire., Ladinsky, Mark S., Hwang, Son-Jong., Guo, Yumei., Zhu, Qiyun., Griffiths, Jessica A., Knight , Rob., Bjorkman, Pamela J., Shapiro, Mikhail G., Geschwind, Daniel H., Holschneider, Daniel P., Fischbach, Michael A., Mazmanian, Sarkis K.
    雑誌名
    Nature
    602
    ページ
    647-653
    2022
    DOI
    10.1038/s41586-022-04396-8
    PMID
    35165440
    Online published
    2022 Feb 14
  • HER3 Augmentation via Blockade of EGFR/AKT Signaling Enhances Anticancer Activity of HER3-Targeting Patritumab Deruxtecan in EGFR-Mutated Non-Small Cell Lung Cancer
    著者
    Yonesaka, Kimio., Tanizaki, Junko., Maenishi, Osamu., Haratani, Koji., Kawakami, Hisato., Tanaka, Kaoru., Hayashi, Hidetoshi., Sakai, Kazuko., Chiba, Yasutaka., Tsuya, Asuka., Goto, Hiroki., Otsuka, Eri., Okida, Hiroaki., Kobayashi, Maki., Yoshimoto, Ryoto., Funabashi, Masanori., Hashimoto, Yuuri., Hirotani, Kenji., Kagari, Takashi., Nishio, Kazuto., Nakagawa, Kazuhiko.
    雑誌名
    Clin Cancer Res .
    28
    ページ
    390-403
    2022
    DOI
    10.1158/1078-0432.CCR-21-3359
    PMID
    34921025
    Online published
    2021 Dec 17
  • Analysis of fluoroquinolone-resistance using MIC determination and homology modelling of ParC of contemporary Mycoplasma genitalium strains
    著者
    Hamasuna, Ryoichi., Hanzawa, Hiroyuki., Moritomo, Ayako., Matsumoto, Masahiro., Aono, Hisami., Tomisaki, Ikko., Akasaka, Takaaki., Fujimoto, Naohiro., SkovJensen, Jørgen.
    雑誌名
    J Infect Chemother
    28
    ページ
    377-383
    2022
    DOI
    10.1016/j.jiac.2021.11.011
    PMID
    34836778
    Online published
    2021 Nov 24
  • Highly sensitive in vitro cytokine release assay incorporating high-density preculture
    著者
    Ito, Shiho., Miwa, Kyoko., Hattori, Chiharu., Aida, Tetsuo., Tsuchiya, Yoshimi., Mori, Kazuhiko.
    雑誌名
    J Immunotoxicol
    18
    ページ
    136-143
    2021
    DOI
    10.1080/1547691X.2021.1984617
    PMID
    34644231
    Online published
    2021 Oct 13
  • Datopotamab Deruxtecan, a Novel TROP2-directed Antibody-drug Conjugate, Demonstrates Potent Antitumor Activity by Efficient Drug Delivery to Tumor Cells
    著者
    Okajima, Daisuke.,Yasuda, Satoru., Maejima, Takanori., Karibe, Tsuyoshi., Sakurai, Ken., Aida, Tetsuo., Toki, Tadashi., Yamaguchi, Junko., Kitamura, Michiko., Kamei, Reiko., Fujitani, Tomomichi., Honda, Tomoyo., Shibutani, Tomoko., Muramatsu, Sumie., Nakada, Takashi., Goto, Riki., Takahashi, Shu., Yamaguchi, Miki., Hamada, Hirofumi., Noguchi, Yutaka., Murakami, Masato., Abe, Yuki., Agatsuma, Toshinori.
    雑誌名
    Mol Cancer Ther
    20
    ページ
    2329-2340
    2021
    DOI
    10.1158/1535-7163.MCT-21-0206
    PMID
    34413126
    Online published
    2021 Aug 19
  • Expanded precision medicine capabilities for strengthening oncology drug development at Daiichi Sankyo
    著者
    Murakami, Masato., Tokui, Taro., Nakamaru, Kenji., Cogswell, John., Ford, Shirin Khambata., Gallant, Gilles.
    雑誌名
    Journal of Precision Medicine
    7
    ページ
    14-19
    2021
    DOI
    https://www.thejournalofprecisionmedicine.com/wp-content/uploads/expanded-precision.pdf
    PMID
    Online published
  • 4-Pyridone-3-carboxylic acid as a benzoic acid bioisostere: Design, synthesis, and evaluation of EP300/CBP histone acetyltransferase inhibitors
    著者
    Kanada, Ryutaro., Suzuki, Takashi., Murata, Takeshi., Miyazaki, Masaki., Shimada, Takashi., Kuroha, Mutsumi., Minami, Megumi., Higuchi, Saito., Tominaga, Yuichi., Naito, Hiroyuki.
    雑誌名
    Bioorg Med Chem Lett
    51
    ページ
    128358
    2021
    DOI
    10.1016/j.bmcl.2021.128358
    PMID
    34534674
    Online published
    2021 Sep 14
  • New biphasic system in side-by-side chambers for testing drug dissolution and permeation in vitro (BiDP system)
    著者
    Masada,Takato., Takagi, Toshihide., Minami, Keiko., Kataoka, Makoto., Takeyama, Shoko., Fujii, Yoshimine., Takahashi, Masayuki., Yamashita, Shinji.
    雑誌名
    Journal of Drug Delivery Science and Technology
    65
    ページ
    102747
    2021
    DOI
    10.1016/j.jddst.2021.102747
    PMID
    Online published
    2021 Jul 24
  • Reforms of regulatory pathways for approval of new antineoplastic drugs in Japan from 2004 to 2019 and accompanying changes in pivotal clinical trial designs
    著者
    Hirai, Takehiro., Suzuki, Asuka., Yamori, Takao., Matsuura, Masaaki.
    雑誌名
    Invest New Drugs
    40
    ページ
    142-150
    2022
    DOI
    10.1007/s10637-021-01165-8
    PMID
    34417913
    Online published
    2021 Aug 21
  • A xanthene derivative, DS20060511, attenuates glucose intolerance by inducing skeletal muscle-specific GLUT4 translocation in mice
    著者
    Furuzono, Shinji., Kubota,Tetsuya., Taura, Junki., Konishi, Masahiro., Naito, Asuka., Tsutsui, Masato., Karasawa, Hiroshi., Kubota, Naoto., Kadowaki, Takashi.
    雑誌名
    Commun Biol
    4
    ページ
    994
    2021
    DOI
    10.1038/s42003-021-02491-6
    PMID
    34417555
    Online published
    2021 Aug 20
  • Novel anti-GARP antibody DS-1055a augments anti-tumor immunity by depleting highly suppressive GARP+ regulatory T cells
    著者
    Satoh, Kazuki., Kobayashi, Yoichi., Fujimaki, Kaori., Hayashi, Shinko., Ishida, Saori., Sugiyama, Daisuke., Sato, Takahiko., Lim, Kyungtaek., Miyamoto, Megumi., Kozuma, Shiho., Kadokura, Michinori., Wakita, Kenichi., Hata, Masato., Hirahara, Kazuki., Amano, Masato., Watanabe, Ichiro., Okamoto, Atsushi., Tuettenberg, Andrea., Jonuleit, Helmut., Tanemura, Atsushi., Maruyama, Shoichi., Agatsuma, Toshinori., Wada, Teiji., Nishikawa, Hiroyoshi.
    雑誌名
    Int Immunol
    33
    ページ
    435-446
    2021
    DOI
    10.1093/intimm/dxab027
    PMID
    34235533
    Online published
    2021 Jun 03
  • Corrigendum to “Syntheses and antimicrobial activities of ogipeptin derivatives” [Bioorg. Med. Chem. Lett. 42 (2021) 128093]
    著者
    Takiguchi, Shingo., Homma, Hidehito., Fujisawa, Tetsunori., Hirota-Takahata, Yuki., Ono, Yasunori., Kizuka, Masaaki., Ishii, Yuki., Yoshimura, Satomichi., Nishi, Takahide.
    雑誌名
    Bioorg Med Chem Lett
    47
    ページ
    128228
    2021
    DOI
    10.1016/j.bmcl.2021.128228
    PMID
    34192636
    Online published
    2021 Jun 27